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Search / Trial NCT06132958

Sacituzumab Tirumotecan (MK-2870) in Post Platinum and Post Immunotherapy Endometrial Cancer (MK-2870-005)

Launched by MERCK SHARP & DOHME LLC · Nov 10, 2023

Trial Information

Current as of June 27, 2025

Recruiting

Keywords

Endometrial Cancer Antibody Drug Conjugate (Adc) Trophoblast Cell Surface Antigen 2 (Trop2)

ClinConnect Summary

This clinical trial is studying a new treatment called MK-2870, also known as sacituzumab tirumotecan, for women with endometrial cancer who have already received certain types of treatments. These women have often undergone platinum-based chemotherapy and immunotherapy, which helps the body's immune system fight cancer. The trial aims to find out if MK-2870 can help patients live longer and keep their cancer from worsening compared to standard chemotherapy.

To be eligible for this study, participants must have a confirmed diagnosis of endometrial cancer or a related type called carcinosarcoma and have evaluable disease. They should have previously been treated with platinum chemotherapy and immunotherapy. If you join the trial, you will receive either the new treatment or standard chemotherapy, and the researchers will monitor your health over time to see how well the treatments work. It's important to note that there are certain conditions that might exclude someone from participating, such as specific types of tumors or previous treatments that could interfere with the study.

Gender

FEMALE

Eligibility criteria

  • The main inclusion and exclusion criteria include but are not limited to the following:
  • Inclusion Criteria:
  • Has a histologically-confirmed diagnosis of endometrial carcinoma or carcinosarcoma.
  • Has radiographically evaluable disease, either measurable or nonmeasurable per response evaluation criteria in solid tumors (RECIST 1.1), as assessed by blinded independent central review (BICR).
  • Has received prior platinum-based chemotherapy and anti-programmed cell death 1 protein (PD-1)/anti- programmed cell death ligand 1 (PD-L1) therapy, either separately or in combination.
  • Exclusion Criteria:
  • Has neuroendocrine tumors or endometrial sarcoma, including stromal sarcoma, leiomyosarcoma, adenosarcoma, or other types of pure sarcomas
  • Has a history of documented severe dry eye syndrome, severe Meibomian gland disease and/or blepharitis, or severe corneal disease that prevents/delays corneal healing
  • Has active inflammatory bowel disease requiring immunosuppressive medication or previous history of inflammatory bowel disease
  • Has had a recurrence of endometrial carcinoma or carcinosarcoma more than \>12 months after completing platinum-based therapy administered in the curative-intent setting without any additional platinum-based therapy received in the recurrent setting. Note: 1) If Immunotherapy-based treatment is administered in the recurrent setting, then platinum rechallenge is not required, regardless of the duration of the platinum-free interval from time of adjuvant therapy 2) For Stage IVb disease, treatment that includes gynecological surgery followed by a platinum-based regimen is NOT considered curative-intent per protocol and does not require platinum rechallenge in the recurrent setting, regardless of the duration of the platinum-free interval
  • Has received more than 3 prior lines of therapy for endometrial carcinoma or carcinosarcoma
  • Has history of (noninfectious) pneumonitis/interstitial lung disease that required steroids or has current pneumonitis/interstitial lung disease
  • Has received prior treatment with single-agent nonplatinum based chemotherapy in the third-line setting
  • Has received prior treatment with a trophoblast cell surface antigen 2 (TROP2)-targeted antibody drug conjugate (ADC) (eg, sacituzumab govitecan)
  • Has received prior treatment with a topoisomerase I inhibitor-containing ADC (eg, sacituzumab govitecan or fam-trastuzumab deruxtecan-nxki)
  • Has previously received both single-agent paclitaxel and single-agent doxorubicin in any setting for prior treatment of endometrial cancer
  • Requires recurrent drainage of effusions (e.g., pleural, ascitic, etc.) within 6 weeks before randomization

About Merck Sharp & Dohme Llc

Merck Sharp & Dohme LLC, a subsidiary of Merck & Co., Inc., is a leading global biopharmaceutical company dedicated to discovering, developing, and delivering innovative medicines and vaccines that address unmet medical needs. With a strong focus on research and development, Merck Sharp & Dohme leverages advanced science and technology to enhance patient outcomes across various therapeutic areas, including oncology, infectious diseases, and cardiovascular health. Committed to ethical practices and regulatory compliance, the company actively engages in clinical trials to advance medical knowledge and improve health care for patients worldwide.

Locations

Columbus, Ohio, United States

Warszawa, Mazowieckie, Poland

Montréal, Quebec, Canada

East Melbourne, Victoria, Australia

Frankston, Victoria, Australia

Haifa, , Israel

Petah Tikva, , Israel

Holon, , Israel

Jerusalem, , Israel

Tel Aviv, , Israel

St Leonards, New South Wales, Australia

Ramat Gan, , Israel

Tel Aviv, , Israel

Seoul, , Korea, Republic Of

Miami Beach, Florida, United States

Madrid, Madrid, Comunidad De, Spain

Washington, District Of Columbia, United States

Shreveport, Louisiana, United States

Santiago, Region M. De Santiago, Chile

Santiago, Region M. De Santiago, Chile

Santiago, Region M. De Santiago, Chile

Seongnam, Kyonggi Do, Korea, Republic Of

Seoul, , Korea, Republic Of

Seoul, , Korea, Republic Of

Hospitalet, Barcelona, Spain

Temuco, Araucania, Chile

Rennes, Ille Et Vilaine, France

Seoul, , Korea, Republic Of

Bialystok, Podlaskie, Poland

Ponce, , Puerto Rico

Fort Wayne, Indiana, United States

Mineola, New York, United States

New York, New York, United States

Montréal, Quebec, Canada

Chambray Les Tours, Centre, France

Plérin, Cotes D Armor, France

Athens, Attiki, Greece

Leiden, Zuid Holland, Netherlands

Stavanger, Rogaland, Norway

Kristiansand, Vest Agder, Norway

Oslo, , Norway

Siedlce, Mazowieckie, Poland

Singapore, Central Singapore, Singapore

Madrid, Madrid, Comunidad De, Spain

Barcelona, , Spain

Chur, Grisons, Switzerland

Mobile, Alabama, United States

Columbus, Georgia, United States

Reno, Nevada, United States

Germantown, Tennessee, United States

Houston, Texas, United States

Buenos Aires, Caba, Argentina

La Rioja, , Argentina

Blacktown, New South Wales, Australia

Innsbruck, Tirol, Austria

Gent, Oost Vlaanderen, Belgium

Namur, , Belgium

Ostrava, Moravskoslezsky Kraj, Czechia

Olomouc, Olomoucky Kraj, Czechia

Praha, Praha 8, Czechia

Aarhus, Midtjylland, Denmark

Tampere, Pirkanmaa, Finland

Kuopio, Pohjois Savo, Finland

Helsinki, Uusimaa, Finland

Besançon, Doubs, France

Lille, Nord Pas De Calais, France

Lyon Cedex08, Rhone Alpes, France

Petah Tikva, , Israel

Kuala Lumpur, , Malaysia

Tromsø, Troms, Norway

Oslo, , Norway

Poznan, Wielkopolskie, Poland

San Juan, , Puerto Rico

San Juan, , Puerto Rico

Stockholm, Stockholms Lan, Sweden

Bellinzona, Ticino, Switzerland

Durham, North Carolina, United States

Ciudad Autónoma De Buenos Aires, Buenos Aires, Argentina

Buenos Aires, Caba, Argentina

Ciudad Autónoma De Buenos Aires, Caba, Argentina

Brisbane, Queensland, Australia

Copenhagen, Hovedstaden, Denmark

Turku, Varsinais Suomi, Finland

Roma, Lazio, Italy

Rozzano, Milano, Italy

Brescia, , Italy

Napoli, , Italy

Torino, , Italy

Cordoba, Andalucia, Spain

Madrid, Madrid, Comunidad De, Spain

Berne, , Switzerland

Truro, England, United Kingdom

London, London, City Of, United Kingdom

Manchester, , United Kingdom

New Haven, Connecticut, United States

Evanston, Illinois, United States

Saint Louis, Missouri, United States

Ciudad Autónoma De Buenos Aires, Buenos Aires, Argentina

Buenos Aires, , Argentina

Leuven, Vlaams Brabant, Belgium

Nový Jiín, Novy Jicin, Czechia

Montpellier, Herault, France

Paris, , France

Milano, , Italy

Valencia, Valenciana, Comunitat, Spain

London, England, United Kingdom

London, Sutton, United Kingdom

Roeselare, West Vlaanderen, Belgium

Joinville, Santa Catarina, Brazil

Chicoutimi, Quebec, Canada

Hidaka, Saitama, Japan

Lund, Skane Lan, Sweden

London, Sutton, United Kingdom

Anchorage, Alaska, United States

Los Angeles, California, United States

San Francisco, California, United States

Orlando, Florida, United States

Hackensack, New Jersey, United States

New York, New York, United States

Fargo, North Dakota, United States

Cincinnati, Ohio, United States

Pittsburgh, Pennsylvania, United States

Sioux Falls, South Dakota, United States

Buenos Aires, , Argentina

Buenos Aires, , Argentina

Sydney, New South Wales, Australia

Wien, , Austria

Gent, Oost Vlaanderen, Belgium

Sao Luis, Maranhao, Brazil

Porto Alegre, Rio Grande Do Sul, Brazil

Sorocaba, Sao Paulo, Brazil

Sao Paulo, , Brazil

Vancouver, British Columbia, Canada

Temuco, Araucania, Chile

Santiago, Region M. De Santiago, Chile

Guangzhou, Guangdong, China

Shantou, Guangdong, China

Zhanjiang, Guangdong, China

Nanning, Guangxi, China

Zhengzhou Shi, Henan, China

Wuhan, Hubei, China

Nanjing, Jiangsu, China

Nanchang, Jiangxi, China

Shanghai, Shanghai, China

Chengdu, Sichuan, China

Urumqi, Xinjiang, China

Hangzhou, Zhejiang, China

Linhai, Zhejiang, China

Wenzhou, Zhejiang, China

Copenhagen, Hovedstaden, Denmark

Bordeaux, Aquitaine, France

Toulouse, Haute Garonne, France

Montpellier, Herault, France

Rennes, Ille Et Vilaine, France

Heilbronn, Baden Wurttemberg, Germany

Patras, Achaia, Greece

Cork, , Ireland

Dublin, , Ireland

Bologna, Emilia Romagna, Italy

Aviano, Friuli Venezia Giulia, Italy

Roma, Lazio, Italy

Milano, Lombardia, Italy

Milan, Lombardia, Italy

Candiolo, Torino, Italy

Reggio Emilia, , Italy

Matsuyama, Ehime, Japan

Kurume, Fukuoka, Japan

Otashi, Gunma, Japan

Tokyo, , Japan

Lembah Pantai, Kuala Lumpur, Malaysia

Oslo, , Norway

Girona, Gerona, Spain

Valencia, Valenciana, Comunitat, Spain

Basel, Basel Stadt, Switzerland

East Sussex, Brighton And Hove, United Kingdom

West Islip, New York, United States

Zhengzhou, Henan, China

Shiwa Gun, Iwate, Japan

Koto, Tokyo, Japan

London, London, City Of, United Kingdom

Worcester, Massachusetts, United States

Philadelphia, Pennsylvania, United States

Willow Grove, Pennsylvania, United States

Rio De Janeiro, , Brazil

Chengdu, Sichuan, China

Urumqi, Xinjiang, China

Kunming, Yunnan, China

Brno, Brno Mesto, Czechia

Marousi, Attiki, Greece

Fukuoka, , Japan

L Hospitalet, Barcelona, Spain

Morristown, New Jersey, United States

Santiago, Region M. De Santiago, Chile

Plerin, Cotes D Armor, France

Dublin, , Ireland

Sapporo, Hokkaido, Japan

Tsukuba, Ibaraki, Japan

Niigata Shi, Niigata, Japan

New Orleans, Louisiana, United States

Providence, Rhode Island, United States

Uberlândia, Minas Gerais, Brazil

Zhengzhou, Henan, China

Wuhan, Hubei, China

Ravensburg, Baden Wurttemberg, Germany

Chuo Ku, Tokyo, Japan

Kagoshima, , Japan

Atlanta, Georgia, United States

Augusta, Georgia, United States

Edgewood, Kentucky, United States

Sao Paulo, , Brazil

Edmonton, Alberta, Canada

Hefei, Anhui, China

Fuzhou, Fujian, China

Haikou, Hainan, China

Linyi, Shandong, China

Tübingen, Baden Wurttemberg, Germany

Osaka, , Japan

Nijmegen, Gelderland, Netherlands

Derby, Derbyshire, United Kingdom

Teaneck, New Jersey, United States

Brooklyn, New York, United States

Montreal, Quebec, Canada

Guangzhou, Guangdong, China

Shanghai, Shanghai, China

Hangzhou, Zhejiang, China

Coyoacan, Distrito Federal, Mexico

London, London, City Of, United Kingdom

Changsha, Hunan, China

Augusta, Georgia, United States

Sao Paulo, , Brazil

Mississauga, Ontario, Canada

Guangzhou, Guangdong, China

Harbin, Heilongjiang, China

Changsha, Hunan, China

Milano, , Italy

Nagoya, Aichi, Japan

Toon, Ehime, Japan

Sunto Gun,, Shizuoka, Japan

Glasgow, Scotland, United Kingdom

West Palm Beach, Florida, United States

Ravensburg, Baden Wurttemberg, Germany

Athens, Attiki, Greece

Tucson, Arizona, United States

Santiago, Region M. De Santiago, Chile

Praha, Praha 2, Czechia

Phoenix, Arizona, United States

San Antonio, Texas, United States

The Woodlands, Texas, United States

Ciudad Autónoma De Buenos Aires, Caba, Argentina

Calgary, Alberta, Canada

Beijing, Beijing, China

Nanchang, Jiangxi, China

Chengdu, Sichuan, China

Wenzhou, Zhejiang, China

Bari, , Italy

Roma, , Italy

Amsterdam, Noord Holland, Netherlands

Stockholm, Stockholms Lan, Sweden

Harbin, Heilongjiang, China

Ravensburg, Baden Wurttemberg, Germany

Wuhan, Hubei, China

Mannheim, Baden Wurttemberg, Germany

Tsukuba, Ibaraki, Japan

Koto, Tokyo, Japan

Shinjuku, Tokyo, Japan

San Pedro Garza Garcia, Nuevo Leon, Mexico

San Pedro Garza García, Nuevo Leon, Mexico

Oaxaca De Juarez, Oaxaca, Mexico

Cordoba, , Spain

Kuala Lumpur, , Malaysia

Mexico City, Distrito Federal, Mexico

Berlin, , Germany

Xiamen, Fujian, China

Munich, Bayern, Germany

Koto, Tokyo, Japan

Shinagawa, Tokyo, Japan

Praha, , Czechia

Nagoya, Aichi, Japan

Los Angeles, California, United States

New York, New York, United States

Columbus, Ohio, United States

Munich, Bayern, Germany

Dresden, Sachsen, Germany

Bologna, Emilia Romagna, Italy

Milan, Lombardia, Italy

Candiolo, Torino, Italy

Napoli, , Italy

Warszawa, Mazowieckie, Poland

Poznan, Wielkopolskie, Poland

Porto Alegre, Rio Grande Do Sul, Brazil

Santiago., Region M. De Santiago, Chile

Kunming, Yunnan, China

Cork, , Ireland

Praha, , Czechia

Praha, , Czechia

Praha, , Czechia

Essen, Nordrhein Westfalen, Germany

Madrid, , Spain

Madrid, , Spain

Madrid, , Spain

Valencia, , Spain

Valencia, , Spain

London, , United Kingdom

London, , United Kingdom

London, , United Kingdom

Patients applied

0 patients applied

Trial Officials

Medical Director

Study Director

Merck Sharp & Dohme LLC

Timeline

First submit

Trial launched

Trial updated

Estimated completion

Not reported