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Search / Trial NCT06629779

A Study to Learn How PF-06821497 (Mevrometostat) Works in Men With Metastatic Castration-resistant Prostate Cancer.

Launched by PFIZER · Sep 27, 2024

Trial Information

Current as of June 27, 2025

Recruiting

Keywords

Mevrometostat Metastatic Castration Resistant Prostate Cancer Pf 06821497 Ezh2 Enhancer Of Zeste Homologue 2 Enzalutamide M Crpc Prostrate Cancer Castrate Resistant Prostate Cancer Prostatecancer Study.Com Efficacy Safety Pharmacokinetics Pharmacodynamics

ClinConnect Summary

This clinical trial is studying a new drug called PF-06821497 (also known as Mevrometostat) to see if it works better when combined with another medication called enzalutamide for men with metastatic castration-resistant prostate cancer (mCRPC). This type of cancer has spread beyond the prostate and does not respond to hormone therapy that lowers testosterone levels. The researchers want to find out if the combination of these two drugs can help patients more than enzalutamide alone, especially for those who haven't received other specific treatments yet.

To participate in this study, men must be at least 18 years old, have a confirmed diagnosis of prostate cancer that has spread, and be receiving hormone therapy to keep testosterone levels low. They should also have progressive disease while on this hormone treatment. However, certain health conditions, recent surgeries, or previous treatments may make someone ineligible. If you join this study, you will receive regular check-ups and monitoring to see how the treatment affects your cancer and overall health. This trial is currently recruiting participants, so if you or someone you know is interested, it's a good opportunity to discuss with a healthcare provider.

Gender

MALE

Eligibility criteria

  • Inclusion Criteria:
  • Histologically or cytologically confirmed adenocarcinoma of the prostate without small cell features.
  • Metastatic disease in bone documented on bone scan, or in soft tissue documented on CT/MRI scan.
  • Progressive disease in the setting of medical or surgical castration.
  • ECOG performance status 0 or 1, with a life expectancy of ≥12 months as assessed by the investigator.
  • Exclusion Criteria:
  • Any medical or psychiatric condition including recent (within the past year) or active suicidal ideation/behavior or laboratory abnormality that make the participant inappropriate for the study.
  • Known history of active inflammatory gastrointestinal disease, chronic diarrhea, or previous gastric resection or lap-band surgery.
  • Clinically significant cardiovascular disease.
  • Known or suspected brain metastasis or active leptomeningeal disease or clinically significant history of seizure.
  • Any history of myelodysplastic syndrome, acute myeloid leukemia, or any other prior malignancy with a few exceptions.
  • * Participants must be treatment naïve at the mCRPC stage, eg, no cytotoxic chemotherapy, radio-ligand therapy (i.e. 177Lu- PSMA-617), CDK4/6 inhibitors, 5-alpha reductase inhibitors for prostate cancer in any setting, androgen receptor signaling inhibitors (ARSi) including enzalutamide, apalutamide, darolutamide, poly ADP-ribose polymerase (PARP) monotherapy or other systemic anti-cancer treatment with the following exceptions:
  • 1. Treatment with first-generation antiandrogen (ADT) agents;
  • 2. Docetaxel treatment is allowed for mCSPC, as long as no signs of failure, or disease progression occurred during treatment or within 3 months of treatment completion.
  • Previous administration with an investigational product (drug or vaccine) within 30 days or 5 half-lives preceding the first dose of study intervention (whichever is longer).
  • Inadequate organ function.

About Pfizer

Pfizer Inc. is a global leader in biopharmaceutical innovation, dedicated to discovering, developing, and delivering advanced therapies that enhance patient outcomes across a wide range of medical conditions. With a rich history of scientific research and a commitment to quality, Pfizer focuses on areas such as oncology, immunology, cardiology, and rare diseases. The company leverages cutting-edge technology and collaborates with healthcare professionals, regulatory bodies, and academic institutions to conduct rigorous clinical trials that ensure the safety and efficacy of its products. Pfizer's mission is to bring breakthroughs that change patients' lives, exemplifying its commitment to health and wellness worldwide.

Locations

Edmonton, Alberta, Canada

Seattle, Washington, United States

Madrid, , Spain

Sapporo, Hokkaido, Japan

Seattle, Washington, United States

Seattle, Washington, United States

Glendale, Arizona, United States

Kashiwa, Chiba, Japan

Sapporo, Hokkaido, Japan

Glasgow, , United Kingdom

Taipei, , Taiwan

Milano, , Italy

Yamagata, , Japan

Taichung, , Taiwan

Tainan, , Taiwan

Hamburg, , Germany

Kaohsiung, , Taiwan

Kobe, Hyogo, Japan

Suita, Osaka, Japan

Patras, , Greece

Seoul, , Korea, Republic Of

Seoul, , Korea, Republic Of

Martin, , Slovakia

Prague, , Czechia

Kanazawa, Ishikawa, Japan

Yokohama, Kanagawa, Japan

Yokosuka, Kanagawa, Japan

Halifax, Nova Scotia, Canada

Seoul, , Korea, Republic Of

Jinan, Shandong, China

Shanghai, Shanghai, China

Nijmegen, Gelderland, Netherlands

Matsuyama, Ehime, Japan

Helsinki, , Finland

Brest, , France

Porto Alegre, Rio Grande Do Sul, Brazil

Goyang Si, , Korea, Republic Of

Fukuoka, , Japan

Xi'an, Shaanxi, China

Taipei, , Taiwan

Beijing, Beijing, China

Ostrava, , Czechia

Pierre Bénite, , France

Changsha, Hunan, China

Zhengzhou, Henan, China

Stockholm, , Sweden

Suzhou, Jiangsu, China

Christchurch, Canterbury, New Zealand

Porto Alegre, Rio Grande Do Sul, Brazil

Chandler, Arizona, United States

Springdale, Arkansas, United States

Myrtle Beach, South Carolina, United States

Wuhan, Hubei, China

Valencia, , Spain

Næstved, , Denmark

Hohhot, Inner Mongolia, China

Quincy, Illinois, United States

Shinjuku Ku, Tokyo, Japan

Osaka, , Japan

Wenzhou, Zhejiang, China

Daegu, , Korea, Republic Of

Xinxiang, Henan, China

Kumamoto, , Japan

Guangzhou, Guangdong, China

Nanjing, Jiangsu, China

Roma, Lazio, Italy

Olomouc, , Czechia

Cremona, , Italy

Qingdao, Shandong, China

Soweto, Gauteng, South Africa

Bratislava, , Slovakia

Calgary, Alberta, Canada

Madrid, , Spain

Nürtingen, , Germany

Oshawa, Ontario, Canada

Omaha, Nebraska, United States

Huai'an, Jiangsu, China

Glendale, Arizona, United States

Chiba Shi, Chiba, Japan

Nantong, Jiangsu, China

Seoul, Jongno Gu, Korea, Republic Of

Yantai, Shandong, China

Beijing, Beijing, China

Olomouc, Olomoucký Kraj, Czechia

Terni, , Italy

Turku, Varsinais Suomi, Finland

Tübingen, , Germany

Fuzhou, Fujian, China

Myrtle Beach, South Carolina, United States

Trencin, , Slovakia

Jiaxing, , China

Seoul, Seoul Teukbyeolsi [Seoul], Korea, Republic Of

Seoul, Seoul Teukbyeolsi [Seoul], Korea, Republic Of

Pierre Bénite, Rhône, France

Gyor, , Hungary

Plovdiv, , Bulgaria

Port Elizabeth, Eastern Cape, South Africa

Montréal, Quebec, Canada

Ankara, , Turkey

Saint Helena, California, United States

Weifang, Shandong, China

Sao Paulo, , Brazil

Rogers, Arkansas, United States

Nürtingen, Baden Württemberg, Germany

Goyang Si, Kyǒnggi Do, Korea, Republic Of

Seoul, Seoul Teukbyeolsi [Seoul], Korea, Republic Of

Reims, , France

Bordeaux, Aquitaine, France

Athens, , Greece

Kraków, Małopolskie, Poland

Buenos Aires, , Argentina

Salisbury, North Carolina, United States

Fayetteville, Arkansas, United States

Verona, , Italy

Xi'an, Shaanxi, China

São José Do Rio Preto, São Paulo, Brazil

Prague, Praha 4, Czechia

Vejle, Syddanmark, Denmark

Tampere, Pirkanmaa, Finland

Tauranga, Bay Of Plenty, New Zealand

Prague, , Czechia

Pretoria, Gauteng, South Africa

Brest, Finistère, France

Trento, , Italy

Torun, Kujawsko Pomorskie, Poland

Patras, Achaḯa, Greece

Chicoutimi, Quebec, Canada

Strasbourg, Alsace, France

Oulu, Pohjois Pohjanmaa, Finland

Athens, Attikí, Greece

Mar Del Plata, Buenos Aires, Argentina

George, Western Cape, South Africa

Pardubice, Pardubický Kraj, Czechia

Gyor, Győr Moson Sopron, Hungary

Daegu, Taegu Kwangyǒkshi, Korea, Republic Of

Madrid, Madrid, Comunidad De, Spain

Capital, Córdoba, Argentina

Wuhu, Anhui, China

Prague, , Czechia

Prague, , Czechia

Næstved, Sjælland, Denmark

Saint Herblain, Loire Atlantique, France

Le Mans, Pays De La Loire, France

Münster, Nordrhein Westfalen, Germany

Valencia, Valenciana, Comunitat, Spain

Blackburn, Blackburn With Darwen, United Kingdom

Myrtle Beach, South Carolina, United States

Tübingen, Baden Württemberg, Germany

Chaidari, Attikí, Greece

Ostrava, Moravskoslezský Kraj, Czechia

Athens, Attikí, Greece

Stockholm, , Sweden

Hwasun, Jeonranamdo, Korea, Republic Of

Roma, Lazio, Italy

Pleven, , Bulgaria

Kuopio, Pohjois Savo, Finland

Santo André, São Paulo, Brazil

Rome, Roma, Italy

Lyon Cedex08, Rhône Alpes, France

Reims, Marne, France

Natal, Rio Grande Do Norte, Brazil

Cheng Du, Sichuan, China

Phoenix, Arizona, United States

Ankara, , Turkey

Kraków, Małopolskie, Poland

Ningbo, Zhejiang, China

Meldola, Emilia Romagna, Italy

Ostrava Poruba, , Czechia

Gabrovo, , Bulgaria

Guilin, Guangxi, China

Cordoba, Córdoba, Argentina

Athens, , Greece

Jung Gu, Taejǒn Kwangyǒkshi, Korea, Republic Of

Santo André, , Brazil

São Paulo, , Brazil

Larissa, Thessalía, Greece

Lublin, Lubelskie, Poland

San Antonio, Texas, United States

Lisle, Illinois, United States

Lisle, Illinois, United States

Westmont, Illinois, United States

Gilbert, Arizona, United States

Mesa, Arizona, United States

Scottsdale, Arizona, United States

Tucson, Arizona, United States

Tucson, Arizona, United States

Myrtle Beach, South Carolina, United States

Cordoba, , Argentina

Piotrków Trybunalski, łódzkie, Poland

Sao Paulo, São Paulo, Brazil

Shantou, Guangdong, China

Hangzhou City, Zhejiang, China

Caba, Buenos Aires, Argentina

Capital Federal, Buenos Aires, Argentina

Hidden Valley Lake, California, United States

Napa, California, United States

Quincy, Illinois, United States

Buenos Aires, , Argentina

Buenos Aires, , Argentina

Jiaxing, Zhejiang/Nanhu, China

Shenyang, , China

Prague, Praha 2, Czechia

Clermont Ferrand, , France

Miskolc, , Hungary

Suita, Osaka, Japan

Saint Grégoire, Ille Et Vilaine, France

Bronx, New York, United States

Stara Zagora, , Bulgaria

Miskolc, Borsod Abaúj Zemplén, Hungary

İstanbul, İ̇stanbul, Turkey

Mar Del Plata, Buenos Aires, Argentina

Piotrków Trybunalski, , Poland

Ostrava Poruba, Moravskoslezský Kraj, Czechia

Kraków, , Poland

Capital, , Argentina

São José Do Rio Preto, , Brazil

Pardubice, , Czechia

Jung Gu, , Korea, Republic Of

Lyon Cedex08, , France

Kraków, , Poland

Wroclaw, , Poland

Larissa, , Greece

Chaidari, , Greece

Fortaleza, , Brazil

İstanbul, , Turkey

Porto Alegre, Rio Grande Do Sul, Brazil

Patients applied

0 patients applied

Trial Officials

Pfizer CT.gov Call Center

Study Director

Pfizer

Timeline

First submit

Trial launched

Trial updated

Estimated completion

Not reported