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Search / Trial NCT02706951

A Study Comparing Upadacitinib (ABT-494) Monotherapy to Methotrexate (MTX) Monotherapy in Adults With Rheumatoid Arthritis (RA) Who Have an Inadequate Response to MTX (SELECT-MONOTHERAPY)

Launched by ABBVIE · Mar 8, 2016

Trial Information

Current as of May 06, 2025

Completed

Keywords

Musculoskeletal Disease Arthritis Joint Disease Anti Inflammatory Agents Antirheumatic Agents Upadacitinib Abt 494

ClinConnect Summary

The study includes a 35-day screening period; a 14-week randomized, double-blind, parallel-group, controlled treatment period (Period 1); a 246-week blinded extension period (Period 2); and a 30-day follow-up visit.

Participants who met eligibility criteria were to be randomized in a 2:2:1:1 ratio to one of four treatment groups:

* Group 1: upadacitinib 30 mg QD (Period 1) → upadacitinib 30 mg QD (Period 2)
* Group 2: upadacitinib 15 mg QD (Period 1) → upadacitinib 15 mg QD (Period 2)
* Group 3: MTX (Period 1) → upadacitinib 30 mg QD (Period 2)
* Group 4: MTX (Period 1) → upadacitinib 15 ...

Gender

ALL

Eligibility criteria

  • Inclusion Criteria:
  • Diagnosis of RA for \>= 3 months.
  • Subjects must have been on oral or parenteral MTX therapy \>= 3 months and on a stable dose for \>= 4 weeks prior to first dose of study drug.
  • Must have discontinued all conventional synthetic disease-modifying anti-rheumatic drugs (csDMARDs) (other than MTX) \>= 4 weeks prior to first dose of study drug.
  • Meets the following minimum disease activity criteria: \>= 6 swollen joints (based on 66 joint counts) and \>= 6 tender joints (based on 68 joint counts) at Screening and Baseline Visits.
  • Exclusion Criteria:
  • Prior exposure to any Janus kinase (JAK) inhibitor (including but not limited to tofacitinib, baricitinib, and filgotinib).
  • Prior exposure to any biological disease-modifying anti-rheumatic drugs (bDMARDs).
  • Current diagnosis of inflammatory joint disease other than RA. Current diagnosis of secondary Sjogren's Syndrome is permitted.

About Abbvie

AbbVie is a global biopharmaceutical company dedicated to developing innovative therapies that address complex health challenges. Founded in 2013 as a spin-off from Abbott Laboratories, AbbVie focuses on key therapeutic areas, including immunology, oncology, neuroscience, and virology. The company is committed to advancing scientific research and delivering groundbreaking treatments that enhance patient outcomes and quality of life. With a robust pipeline and a strong emphasis on collaboration, AbbVie strives to transform the future of medicine through its commitment to clinical excellence and patient-centered approaches.

Locations

Huntsville, Alabama, United States

Mobile, Alabama, United States

Gilbert, Arizona, United States

Phoenix, Arizona, United States

Tucson, Arizona, United States

Jonesboro, Arkansas, United States

Hemet, California, United States

Colorado Springs, Colorado, United States

Fort Lauderdale, Florida, United States

Miami Springs, Florida, United States

Pinellas Park, Florida, United States

Sarasota, Florida, United States

Tamarac, Florida, United States

Tampa, Florida, United States

Tampa, Florida, United States

Tampa, Florida, United States

Tampa, Florida, United States

Tampa, Florida, United States

Decatur, Georgia, United States

Chicago, Illinois, United States

Wichita, Kansas, United States

Baton Rouge, Louisiana, United States

Monroe, Louisiana, United States

Shreveport, Louisiana, United States

Mansfield, Massachusetts, United States

Omaha, Nebraska, United States

Lebanon, New Hampshire, United States

Albuquerque, New Mexico, United States

Las Cruces, New Mexico, United States

New Bern, North Carolina, United States

Vandalia, Ohio, United States

Oklahoma City, Oklahoma, United States

Tulsa, Oklahoma, United States

Greenville, South Carolina, United States

Nashville, Tennessee, United States

Austin, Texas, United States

Beaumont, Texas, United States

Carrollton, Texas, United States

College Station, Texas, United States

Corpus Christi, Texas, United States

Houston, Texas, United States

Houston, Texas, United States

Houston, Texas, United States

Lufkin, Texas, United States

Mesquite, Texas, United States

San Antonio, Texas, United States

San Marcos, Texas, United States

The Woodlands, Texas, United States

Tomball, Texas, United States

Waco, Texas, United States

Chesapeake, Virginia, United States

Franklin, Wisconsin, United States

Buenos Aires, , Argentina

Buenos Aires, , Argentina

Buenos Aires, , Argentina

Buenos Aires, , Argentina

Salta, , Argentina

Santa Fe, , Argentina

Camperdown, New South Wales, Australia

Wien, , Austria

Aalst, Oost Vlaanderen, Belgium

Genk, , Belgium

Sofia, , Bulgaria

Sofia, , Bulgaria

Concepcion, , Chile

Puerto Varas, , Chile

Santiago, , Chile

Olomouc, Olomoucky Kraj, Czechia

Prague 4, Praha 4, Czechia

Prague 4, Praha 4, Czechia

Breclav, , Czechia

Uherské Hradište, , Czechia

Tartu, Tartumaa, Estonia

Tallinn, , Estonia

Athens, , Greece

Veszprém, Veszprem, Hungary

Budapest, , Hungary

Kistarcsa, , Hungary

Szekesfehervar, , Hungary

Ashkelon, , Israel

Haifa, , Israel

Haifa, , Israel

Ramat Gan, , Israel

Catanzaro, Calabria, Italy

Verona, , Italy

Fukuoka Shi, Fukuoka, Japan

Fukuoka Shi, Fukuoka, Japan

Fukuoka Shi, Fukuoka, Japan

Iizuka Shi, Fukuoka, Japan

Takasaki, Gunma, Japan

Kochi Shi, Kochi, Japan

Kumamoto Shi, Kumamoto, Japan

Kumamoto Shi, Kumamoto, Japan

Nagasaki Shi, Nagasaki, Japan

Sasebo City, Nagasaki, Japan

Osaka Shi, Osaka, Japan

Hamamatsu, , Japan

Hyuga, , Japan

Nishimura, , Japan

Sanuki, , Japan

Sapporo, , Japan

Sapporo, , Japan

Shunan, , Japan

Takaoka, , Japan

Tokyo, , Japan

Yotsukaido, , Japan

Monterrey, Nuevo Leon, Mexico

Mexico City, , Mexico

Wrocław, Dolnoslaskie, Poland

Lublin, Lubelskie, Poland

Warszawa, Mazowieckie, Poland

Białystok, Podlaskie, Poland

Gdansk, Pomorskie, Poland

Elblag, Warminsko Mazurskie, Poland

Poznań, Wielkopolskie, Poland

Lisbon, Lisboa, Portugal

Vila Nova De Gaia, Porto, Portugal

Lisboa, , Portugal

Porto, , Portugal

Carolina, , Puerto Rico

Ponce, , Puerto Rico

Ploiesti, , Romania

Moscow, Moskva, Russian Federation

Novosibirsk, Novosibirskaya Oblast, Russian Federation

Perm, Permskiy Kray, Russian Federation

Tver, Tverskaya Oblast, Russian Federation

Ivanovo, , Russian Federation

Moscow, , Russian Federation

Nizhnij Novgorod, , Russian Federation

Orenburg, , Russian Federation

Petrozavodsk, , Russian Federation

Samara, , Russian Federation

Ufa, , Russian Federation

Yaroslavl, , Russian Federation

Belgrade, Beograd, Serbia

Belgrade, Beograd, Serbia

Belgrade, Beograd, Serbia

Novi Sad, Vojvodina, Serbia

Johannesburg, Gauteng, South Africa

Pretoria, Gauteng, South Africa

Cape Town, Western Cape, South Africa

Cape Town, Western Cape, South Africa

Barcelona, , Spain

Barcelona, , Spain

Sevilla, , Spain

Sevilla, , Spain

Valencia, , Spain

Osmangazi, Bursa, Turkey

Lviv, Lvivska Oblast, Ukraine

Vinnytsia, Vinnytska Oblast, Ukraine

Ivano Frankivsk, , Ukraine

Kiev, , Ukraine

Zaporizhia, , Ukraine

Patients applied

0 patients applied

Trial Officials

AbbVie Inc.

Study Director

AbbVie

Timeline

First submit

Trial launched

Trial updated

Estimated completion

Not reported

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