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Search / Trial NCT04607421

A Study of Encorafenib Plus Cetuximab With or Without Chemotherapy in People With Previously Untreated Metastatic Colorectal Cancer

Launched by PFIZER · Oct 22, 2020

Trial Information

Current as of May 20, 2025

Active, not recruiting

Keywords

Colorectal Cancer Colon Cancer Rectal Cancer Colorectal Neoplasms Intestinal Cancer Intestinal Neoplasms Gastrointestinal Cancer Gastrointestinal Neoplasms Digestive System Cancer Digestive System Neoplasms Digestive System Diseases Gastrointestinal Diseases Colonic Diseases Intestinal Diseases Rectal Diseases Breakwater Study

ClinConnect Summary

This clinical trial is studying the effectiveness of two medications, encorafenib and cetuximab, either on their own or combined with standard chemotherapy, for treating a specific type of colorectal cancer that has spread to other parts of the body. This cancer must have a particular genetic change called the "BRAF V600E mutation," and patients must not have received any previous treatments for their cancer. Participants will be assigned to one of three treatment groups: one group will receive encorafenib and cetuximab, another group will receive those same medications along with chemotherapy, and the last group will receive chemotherapy alone.

To be eligible for this study, participants should be at least 16 years old, have confirmed stage IV colorectal cancer with the BRAF mutation, and have measurable disease. They should not have received more than one previous treatment for metastatic cancer. Throughout the study, which may last up to three years, the research team will closely monitor how each participant responds to their assigned treatment. It's important to note that the study is currently active but not recruiting new participants.

Gender

ALL

Eligibility criteria

  • Inclusion Criteria:
  • Safety Lead-In = Male/female ≥ 18 years old
  • Phase 3 and Cohort 3: Male/female ≥ 16 years old (where permitted locally)
  • Histologically or cytologically confirmed Stage IV CRC that contains BRAF V600E mutation
  • Prior systemic treatment in metastatic setting: 0-1 regimens for Safety Lead In; none for Phase 3 and Cohort 3. (Note: Prior adjuvant or neoadjuvant therapy considered metastatic treatment if relapse/metastasis \< 6 month from end of adj/neoadjuvant treatment )
  • Measurable disease (Phase 3 and Cohort 3)/ Measurable or evaluable disease (Safety Lead-in)
  • ECOG PS 0-1
  • Adequate organ function
  • Exclusion Criteria:
  • Tumors that are locally confirmed or unknown MSI-H or dMMR unless participant is ineligible to receive immune checkpoint inhibitors due to a pre-existing medical condition
  • Active bacterial or viral infections in 2 weeks prior to starting dosing
  • Symptomatic brain metastases

About Pfizer

Pfizer Inc. is a global leader in biopharmaceutical innovation, dedicated to discovering, developing, and delivering advanced therapies that enhance patient outcomes across a wide range of medical conditions. With a rich history of scientific research and a commitment to quality, Pfizer focuses on areas such as oncology, immunology, cardiology, and rare diseases. The company leverages cutting-edge technology and collaborates with healthcare professionals, regulatory bodies, and academic institutions to conduct rigorous clinical trials that ensure the safety and efficacy of its products. Pfizer's mission is to bring breakthroughs that change patients' lives, exemplifying its commitment to health and wellness worldwide.

Locations

Rochester, Minnesota, United States

Ann Arbor, Michigan, United States

Rochester, Minnesota, United States

Saint Louis, Missouri, United States

Brussels, , Belgium

Copenhagen, , Denmark

Edmonton, Alberta, Canada

Calgary, Alberta, Canada

Los Angeles, California, United States

New Orleans, Louisiana, United States

New York, New York, United States

Liverpool, New South Wales, Australia

Madrid, , Spain

Valencia, , Spain

Miami Beach, Florida, United States

Zaragoza, , Spain

Portland, Oregon, United States

Nashville, Tennessee, United States

Seattle, Washington, United States

Portland, Oregon, United States

Washington, District Of Columbia, United States

Los Angeles, California, United States

Washington, District Of Columbia, United States

Cleveland, Ohio, United States

Seattle, Washington, United States

Sapporo, Hokkaido, Japan

Nashville, Tennessee, United States

Charlotte, North Carolina, United States

Chicago, Illinois, United States

Miami, Florida, United States

Miami, Florida, United States

Orlando, Florida, United States

Miami Beach, Florida, United States

Toronto, Ontario, Canada

Los Angeles, California, United States

Richmond, Virginia, United States

Pittsburgh, Pennsylvania, United States

Los Angeles, California, United States

Miami, Florida, United States

Melbourne, Victoria, Australia

Woolloongabba, Queensland, Australia

Phoenix, Arizona, United States

Montreal, Quebec, Canada

Taichung, , Taiwan

Ann Arbor, Michigan, United States

Houston, Texas, United States

Valencia, , Spain

Jacksonville, Florida, United States

Pretoria, , South Africa

Richmond, Virginia, United States

Houston, Texas, United States

Heidelberg, Victoria, Australia

Mumbai, Maharashtra, India

Odense C, , Denmark

Elche, Alicante, Spain

Helsinki, , Finland

Nagoya, Aichi, Japan

Kashiwa, Chiba, Japan

Chuo Ku, Tokyo, Japan

Herlev, , Denmark

Dresden, , Germany

Madrid, , Spain

Taipei, , Taiwan

Taipei, , Taiwan

Turku, , Finland

Savannah, Georgia, United States

Oulu, , Finland

Taichung, , Taiwan

New York, New York, United States

Sevilla, , Spain

Leuven, , Belgium

Kaohsiung, , Taiwan

Leuven, , Belgium

Seoul, , Korea, Republic Of

Savannah, Georgia, United States

Seoul, , Korea, Republic Of

Barcelona, , Spain

Suita, Osaka, Japan

Hannover, Niedersachsen, Germany

Porto Alegre, Rio Grande Do Sul, Brazil

Pori, , Finland

Incheon, , Korea, Republic Of

Tainan, , Taiwan

Leipzig, Sachsen, Germany

Seoul, , Korea, Republic Of

Seoul, , Korea, Republic Of

Seoul, , Korea, Republic Of

Auckland, , New Zealand

Bratislava, , Slovakia

Barcelona, , Spain

Melbourne, Victoria, Australia

Madrid, , Spain

Kanazawa, Ishikawa, Japan

Busan, , Korea, Republic Of

Herston, Queensland, Australia

Birmingham, , United Kingdom

Antwerpen, , Belgium

Beijing, Beijing, China

Guangzhou, Guangdong, China

Beijing, , China

Guangzhou, , China

Seoul, , Korea, Republic Of

Berkeley Heights, New Jersey, United States

Saint Louis, Missouri, United States

Los Angeles, California, United States

Orlando, Florida, United States

Osakasayama, Osaka, Japan

Beijing, , China

Charlotte, North Carolina, United States

Praha 5, , Czechia

Matsuyama, Ehime, Japan

Taoyuan, , Taiwan

Berlin, , Germany

Utrecht, , Netherlands

Wexford, Pennsylvania, United States

Eindhoven, Noord Brabant, Netherlands

Camperdown, New South Wales, Australia

Hradec Kralove, , Czechia

Adelaide, South Australia, Australia

Goyang Si, , Korea, Republic Of

Incheon, , Korea, Republic Of

Sutton, Surrey, United Kingdom

Fukuoka, , Japan

London, , United Kingdom

Taipei, , Taiwan

Orlando, Florida, United States

Ivano Frankivsk, , Ukraine

Pune, Maharashtra, India

Zhengzhou, Henan, China

Daegu, , Korea, Republic Of

Columbus, Ohio, United States

Milano, , Italy

Commack, New York, United States

Changsha, Hunan, China

Maastricht, , Netherlands

Richmond, Virginia, United States

Hefei, , China

Los Angeles, California, United States

Seoul, , Korea, Republic Of

Fuzhou, Fujian, China

Charleroi, Hainaut, Belgium

Creve Coeur, Missouri, United States

Tampere, , Finland

Changsha, , China

Beijing, Beijing, China

Pune, Maharashtra, India

Poprad, , Slovakia

Los Angeles, California, United States

Charlotte, North Carolina, United States

Aalborg, , Denmark

Madison, Wisconsin, United States

Brescia, , Italy

Melbourne, Victoria, Australia

Johannesburg, Gauteng, South Africa

Nashville, Tennessee, United States

Shenyang, , China

Plovdiv, , Bulgaria

Changsha, Hunan, China

Savannah, Georgia, United States

Cordoba, , Argentina

Nagaizumi, Shizuoka, Japan

Hannover, Lower Saxony, Germany

Guangzhou, Guangdong, China

Columbus, Ohio, United States

London, , United Kingdom

Milwaukee, Wisconsin, United States

Berlin, , Germany

Yokohama, Kanagawa, Japan

Saint Louis, Missouri, United States

Herlev, , Denmark

Billings, Montana, United States

Tianjin, , China

Koto Ku, Tokyo, Japan

Daegu, , Korea, Republic Of

Basking Ridge, New Jersey, United States

Columbus, Ohio, United States

New Lenox, Illinois, United States

Los Angeles, California, United States

Goyang Si, Gyeonggi Do, Korea, Republic Of

St Leonards, New South Wales, Australia

Olomouc, , Czechia

Saint Peters, Missouri, United States

Gdansk, , Poland

Barretos, Sp, Brazil

Taipei, , Taiwan

Bergen, Hordaland, Norway

Portland, Oregon, United States

Santo Andre, Sp, Brazil

Saransk, Republic Of Mordovia, Russian Federation

Kharkiv, , Ukraine

Padova, , Italy

Kosice, , Slovakia

Clayton, Victoria, Australia

Guangzhou, , China

Concord, North Carolina, United States

Omsk, , Russian Federation

Tainan, , Taiwan

Hamburg, , Germany

Chiba Shi, Chiba, Japan

London, , United Kingdom

São José Do Rio Preto, , Brazil

Brzozow, , Poland

Shanghai, Shanghai, China

Jinan, Shandong, China

Beijing, Beijing, China

Fort Lauderdale, Florida, United States

Panagyurishte, Pazardzhik, Bulgaria

Plovdiv, , Bulgaria

Lajeado, Rio Grande Do Sul, Brazil

Orenburg, , Russian Federation

Plantation, Florida, United States

St. Petersburg, , Russian Federation

Santo Andre, Sp, Brazil

Montvale, New Jersey, United States

Cordoba, , Argentina

Harrison, New York, United States

Middletown, New Jersey, United States

Florham Park, New Jersey, United States

New Delhi, Delhi, India

London, Ontario, Canada

Pushkin, Saint Petersburg, Russian Federation

Yaroslavl, , Russian Federation

San Giovanni Rotondo, Foggia, Italy

Wuhan, Hubei, China

Shanghai, Shanghai, China

Maastricht, Limburg, Netherlands

Orland Park, Illinois, United States

Hamburg, , Germany

Hamburg, , Germany

Oslo, , Norway

Oldenburg, , Germany

Uniondale, New York, United States

Wilrijk, , Belgium

Nanning, Guangxi, China

Milan, Milano, Italy

Chongqing, Chongqing, China

Jeonnam, , Korea, Republic Of

Charlotte, North Carolina, United States

Charlotte, North Carolina, United States

Monroe, North Carolina, United States

Seoul, Seoul Teukbyeolsi [Seoul], Korea, Republic Of

Seoul, Seoul Teukbyeolsi [Seoul], Korea, Republic Of

Chicago, Illinois, United States

Chicago, Illinois, United States

Flossmoor, Illinois, United States

Harvey, Illinois, United States

Tinley Park, Illinois, United States

Florissant, Missouri, United States

Rochester, Minnesota, United States

Chelyabinsk, , Russian Federation

Amsterdam, , Netherlands

Shenyang, Liaoning, China

Plovdiv, , Bulgaria

Kyiv, , Ukraine

Portland, Oregon, United States

Portland, Oregon, United States

Port Elizabeth, Eastern Cape, South Africa

Saint Petersburg, , Russian Federation

Saint Petersburg, , Russian Federation

Chongqing, Chongqing, China

Kortrijk, West Vlaanderen, Belgium

Nanjing, Jiangsu, China

Scottsdale, Arizona, United States

Dnipro, , Ukraine

Gabrovo, , Bulgaria

Västerås, , Sweden

Plantation, Florida, United States

Hefei, Anhui, China

Ina Machi, Saitama, Japan

New Delhi, Delhi, India

Kaluga, , Russian Federation

Córdoba, , Argentina

Copenhagen, Region Hovedstaden, Denmark

London, , United Kingdom

Takatsuki, Osaka, Japan

Tokyo, , Japan

Pittsburgh, Pennsylvania, United States

Kharkiv, , Ukraine

St Leonards, New South Wales, Australia

Saint Petersburg, , Russian Federation

New York, New York, United States

Saint Petersburg, , Russian Federation

Ivano Frankivsk, , Ukraine

Praha 8, , Czechia

Concord, North Carolina, United States

Banska Bystrica, , Slovakia

Jaipur, Rajasthan, India

Gilly, Hainaut, Belgium

Phoenix, Arizona, United States

Beverly Hills, California, United States

Pasadena, California, United States

Torrance, California, United States

Aventura, Florida, United States

Coral Gables, Florida, United States

Savannah, Georgia, United States

Savannah, Georgia, United States

New Orleans, Louisiana, United States

Billings, Montana, United States

Omaha, Nebraska, United States

Omaha, Nebraska, United States

Papillion, Nebraska, United States

Babylon, New York, United States

Bronx, New York, United States

New York, New York, United States

Patchogue, New York, United States

Port Jefferson Station, New York, United States

Riverhead, New York, United States

Charlotte, North Carolina, United States

Charlotte, North Carolina, United States

Charlotte, North Carolina, United States

Columbus, Ohio, United States

Oklahoma City, Oklahoma, United States

Portland, Oregon, United States

Jefferson Hills, Pennsylvania, United States

Monroeville, Pennsylvania, United States

Pittsburgh, Pennsylvania, United States

Pittsburgh, Pennsylvania, United States

Pittsburgh, Pennsylvania, United States

Clarksville, Tennessee, United States

Franklin, Tennessee, United States

Gallatin, Tennessee, United States

Germantown, Tennessee, United States

Hendersonville, Tennessee, United States

Hermitage, Tennessee, United States

La Vergne, Tennessee, United States

Lebanon, Tennessee, United States

Memphis, Tennessee, United States

Murfreesboro, Tennessee, United States

Nashville, Tennessee, United States

Nashville, Tennessee, United States

Nashville, Tennessee, United States

Nashville, Tennessee, United States

Nashville, Tennessee, United States

Nashville, Tennessee, United States

Smyrna, Tennessee, United States

Richmond, Virginia, United States

San Miguel De Tucumán, Tucumán, Argentina

Tucuman, Tucumán, Argentina

Ciudad Autónoma De Buenos Aires, , Argentina

Mount Kuring Gai, New South Wales, Australia

Newtown, New South Wales, Australia

St Leonards, New South Wales, Australia

Brussels, Bruxelles Capitale, Région De, Belgium

Brussels, Bruxelles Capitale, Région De, Belgium

Verviers, Liège, Belgium

Liège, , Belgium

Rio De Janeiro, Rj, Brazil

Rio De Janeiro, Rj, Brazil

Blumenau, Santa Catarina, Brazil

Itajaí, Santa Catarina, Brazil

Santo André, Sp, Brazil

Barretos, São Paulo, Brazil

Sao Jose Do Rio Preto, São Paulo, Brazil

São José Do Rio Preto, São Paulo, Brazil

Sofia, , Bulgaria

Sofia, , Bulgaria

Sofia, , Bulgaria

Kingston, Ontario, Canada

Laval, Quebec, Canada

Fuzhou, Fujian, China

Qingdao, Shandong, China

Chengdu, Sichuan, China

Kunming, Yunnan, China

Hangzhou, Zhejiang, China

Shanghai, , China

Brno, Brno Město, Czechia

Hradec Kralove, Hradec Králové, Czechia

Prague, Praha 4, Czechia

Aalborg, Nordjylland, Denmark

Vejle, Syddanmark, Denmark

Vejle, Syddanmark, Denmark

Helsinki, Nyland, Finland

Tampere, Pirkanmaa, Finland

Muenchen, Bayern, Germany

Frankfurt, Hessen, Germany

Berlin Charlottenburg, , Germany

Berlin, , Germany

Berlin, , Germany

Dresden, , Germany

Thane, Maharashtra, India

Jaipur, Rajasthan, India

Monserrato (Ca), Cagliari, Italy

Candiolo, Torino, Italy

Orbassano, Torino, Italy

Napoli, , Italy

Reggio Emilia, , Italy

Kawasaki, Kanagawa, Japan

Nagoya, Nagoya, Aichi, Japan

Osaka Shi, Osaka, Japan

Hidaka City, Saitama, Japan

Osaka, , Japan

Daegu, Taegu Kwangyǒkshi, Korea, Republic Of

Jeonnam, , Korea, Republic Of

Monterrey, Nuevo Leon, Mexico

Oaxaca, , Mexico

Amsterdam, Noord Holland, Netherlands

Den Haag, Zuid Holland, Netherlands

Den Haag, , Netherlands

Leidschendam, , Netherlands

Tauranga, Bay Of Plenty, New Zealand

Stavanger, Rogaland, Norway

Trondheim, Sør Trøndelag, Norway

Kristiansand, Vest Agder, Norway

Oslo, , Norway

Konin, Wielkopolskie, Poland

Brzozow, , Poland

Bytom, , Poland

Gdansk, , Poland

Bytom, śląskie, Poland

Nalchik, Kabardino Balkarian Republic, Russian Federation

Moscow, , Russian Federation

Ufa, , Russian Federation

Yaroslavl, , Russian Federation

Yaroslav, , Russian Federation

Bratislava, , Slovakia

Rondebosch, Cape Town, South Africa

Pretoria, Gauteng, South Africa

Cape Town, Western Cape, South Africa

Cape Town, Western Cape, South Africa

Santiago De Compostela, A Coruña, Spain

Hospitalet De Llobregat, Barcelona, Spain

Solna, Stockholms Län [Se 01], Sweden

Uppsala, Uppsala Län [Se 03], Sweden

Umeå, Västerbottens Län [Se 24], Sweden

Göteborg, Västra Götalands Län [Se14], Sweden

Pliuty Village, Kyiv Region, Obuhovskiy District, Ukraine

Ivano Frankivsk, , Ukraine

Kryvyi Rih, , Ukraine

Kyiv, , Ukraine

Zaporizhzhia, , Ukraine

Newcastle Upon Tyne, High Heaton, United Kingdom

Oxford, , United Kingdom

Charleroi, Hainaut, Belgium

Parktown, Johannesburg, Gauteng, South Africa

Jinan, Shandong, China

Copenhagen, Hovedstaden, Denmark

Daegu, Taegu Kwangyǒkshi, Korea, Republic Of

Cleveland, Ohio, United States

Sao Paulo, Sp, Brazil

São Paulo, Sp, Brazil

Hefei, Anhui, China

Leidschendam, Zuid Holland, Netherlands

Auckland, , New Zealand

Santo Andre, Sp, Brazil

Blumenau, Santa Catarina, Brazil

Sevilla, Andalucía, Spain

Columbus, Ohio, United States

Richmond, Virginia, United States

Santo Andre, Sp, Brazil

Parktown, Gauteng, South Africa

Johannesburg, , South Africa

Santo Andre, Sp, Brazil

Calgary, Alberta, Canada

Padova, Veneto, Italy

Calgary, Alberta, Canada

Patients applied

0 patients applied

Trial Officials

Pfizer CT.gov Call Center

Study Director

Pfizer

Timeline

First submit

Trial launched

Trial updated

Estimated completion

Not reported

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